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RR-11a analog
CAS No. 685543-66-2
RR-11a analog ( aza-peptide Michael acceptor, 7a )
产品货号. M26423 CAS No. 685543-66-2
RR-11a analog is a potent and selective asparaginyl endopeptidases (AE) (Legumain) inhibitors(IC50 values of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥3686 | 有现货 |
|
| 10MG | ￥5087 | 有现货 |
|
| 25MG | ￥9396 | 有现货 |
|
| 50MG | ￥16038 | 有现货 |
|
| 100MG | ￥23409 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称RR-11a analog
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述RR-11a analog is a potent and selective asparaginyl endopeptidases (AE) (Legumain) inhibitors(IC50 values of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively).
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产品描述RR-11a analog is a potent and selective asparaginyl endopeptidases (AE) (Legumain) inhibitors(IC50 values of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively).(In Vivo):RR-11a analog shows a t1/2 of 3-10 min.
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同义词aza-peptide Michael acceptor, 7a
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通路Others
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靶点Other Targets
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受体Ligands for Target Protein for PROTAC
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研究领域——
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适应症——
化学信息
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CAS Number685543-66-2
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分子量491.5
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分子式C22H29N5O8
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纯度>98% (HPLC)
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溶解度——
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SMILESCCOC(=O)\C=C\C(=O)N(CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OCc1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Peng ZH, et al. Spacer length impacts the efficacy of targeted docetaxel conjugates in prostate-specific membrane antigen expressing prostate cancer. J Drug Target. 2013 Dec;21(10):968-80.
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